Online Purchasing Account You are logged on as Guest. LoginRegister a New AccountShopping cart (Empty)
United States 


HDAC inhibitor
BML-GR362-0100 100 µg 102.00 USD
BML-GR362-0500 500 µg 419.00 USD
Do you need bulk/larger quantities?
Tubacin (tubulin acetylation inducer) is a highly potent and selective, reversible, cell-permeable inhibitor of HDAC6 (IC50=0.004µM). IC50's for the other HDACs are 1000-fold higher, making tubacin both more selective and more potent than Tubastatin A, which also inhibits HDAC8. Concentration in cell culture experiments typically ranges from 2-50µM.

Product Specification

Alternative Name:N-(4-{(2R,4R,6S)-4-{[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanyl]methyl}-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl}phenyl)-N'-hydroxyoctanediamide
Purity:≥96% (ELSD)
Appearance:White solid.
Solubility:Soluble in DMSO (10 mg/ml).
Shipping:Shipped on Dry Ice
Short Term Storage:-20°C
Long Term Storage:-80°C
Use/Stability:Stable for at least 1 year after receipt when stored at -80°C.
BML-GR362 Structure
Please mouse over
BML-GR362 Structure

Product Literature References

LC3A Silencing Hinders Aggresome Vimentin Cage Clearance in Primary Choroid Plexus Carcinoma: M. Nassar, et al.; Sci. Rep. 7, 8022 (2017), Application(s): Measurement of cell index against different concentration, Abstract; Full Text
Rational design and simple chemistry yield a superior, neuroprotective HDAC6 inhibitor, Tubastatin A: K.V. Butler, et al.; J. Am. Chem. Soc. 370, 10842 (2010), Abstract;
Selective inhibition of histone deacetylase 6 (HDAC6) induces DNA damage and sensitizes transformed cells to anticancer agents: M. Namdar, et al.; Proc. Natl. Acad. Sci. USA 107, 20003 (2010), Abstract; Full Text
Tubacin kills Epstein-Barr virus (EBV)-Burkitt lymphoma cells by inducing reactive oxygen species and EBV lymphoblastoid cells by inducing apoptosis: J. Kawada, et al.; J. Biol. Chem. 284, 17102 (2009), Abstract; Full Text
Histone deacetylase 6 interacts with the microtubule-associated protein tau: H. Ding, et al.; J. Neurochem. 106, 2119 (2008), Abstract; Full Text
Domain-selective small-molecule inhibitor of histone deacetylase 6 (HDAC6)-mediated tubulin deacetylation: S.J. Haggarty, et al.; Proc. Natl. Acad. Sci. USA 100, 4389 (2003), Abstract; Full Text
Multidimensional chemical genetic analysis of diversity-oriented synthesis-derived deacetylase inhibitors using cell-based assays: S.J. Haggarty, et al.; Chem. Biol. 10, 383 (2003), Abstract;
Structural biasing elements for in-cell histone deacetylase paralog selectivity: J.C. Wong, et al.; J. Am. Chem. Soc. 125, 5586 (2003), Abstract;
Synthesis of 7200 small molecules based on a substructural analysis of the histone deacetylase inhibitors trichostatin and trapoxin: S.M. Sternson, et al.; Org. Lett. 3, 4239 (2001), Abstract;

Related Products

HDAC6 (human), (recombinant) (His-tag) 

Highly active
Produced in insect cells. Produced in a baculovirus expression system. | Print as PDF
BML-SE508-0050 50 µg 445.00 USD
Do you need bulk/larger quantities?

FLUOR DE LYS® HDAC6 fluorometric drug discovery kit 

Fluorescent detection, HTS, Activity assay, Cell-based assays | Print as PDF
BML-AK516-0001 96 wells 689.00 USD
Do you need bulk/larger quantities?


HDAC inhibitor
Synthetic., ≥98% (HPLC) | Print as PDF
BML-GR363-0100 100 µg 79.00 USD
BML-GR363-0500 500 µg 318.00 USD
Do you need bulk/larger quantities?

Product Toolbox


Certificate of Analysis


By target:
By biological activity:
HDAC Inhibitor
HDAC6 Inhibitor
By catalog section:


Technical Service
Customer Service

Related Literature

Stem Cells
Stem Cells
Download as PDF

Download as PDF

All new literature pieces

Recommend this page

For Research Use Only. Not for use in diagnostic procedures.
Keep in touch

©2019 Enzo Life Sciences, Inc.,