Irreversible inhibitor of γ-glutamyl transpeptidase (GGT) ID50 = 0.54 mM. Inhibits the enzymatic conversion of leukotriene C4 to leukotriene D4. Displays antitumor and anti-metastatic activity. Blocks H. Pylori GGT-induced T-cell inhibition. Inhibits bioactivation/release of nitric oxide from GSNO.
Product Details
| Alternative Name: | U-42126, AT-125 |
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| Formula: | C5H7ClN2O3 |
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| MW: | 178.6 |
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| CAS: | 42228-92-2 |
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| Purity: | ≥98% (HPLC) |
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| Appearance: | White solid. |
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| Solubility: | Soluble in water (max. 18mg/ml). |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | -20°C |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
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