Potent and selective inhibitor of protein kinase C (PKC).
Product Details
| Formula: | C23H20N4O2 |
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| MW: | 384.4 |
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| Purity: | ≥98% |
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| Identity: | Determined by NMR. |
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| Appearance: | Red solid. |
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| Solubility: | Soluble in methanol or DMSO. |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | -20°C |
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| Handling: | Protect from light. |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Proteome-wide identification of cellular targets affected by bisindolylmaleimide-type protein kinase C inhibitors: D. Brehmer, et al.; Mol. Cell Proteomics
3, 490 (2004),
Abstract;
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Protein kinase C inhibitors; structure-activity relationships in K252c- related compounds: S. Fabre and M. Prudhomme; Bioorg. Med. Chem.
1, 193 (1993),
Abstract;
Inhibitors of protein kinase C. 1. 2,3-Bisarylmaleimides: P.D. Davis, et al.; J. Med. Chem.
35, 177 (1992),
Abstract;
The bisindolylmaleimide GF 109203X is a potent and selective inhibitor of protein kinase C: D. Toullec, et al.; J. Biol. Chem.
266, 15771 (1991),
Abstract;
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