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PGP-4008

P-glycoprotein inhibitor
 
ALX-270-290-M002 2 mg 115.00 USD
 
ALX-270-290-M010 10 mg 372.00 USD
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Selective P-glycoprotein (Pgp) inhibitor. Effectively reverses Pgp mediated drug resistance in NCI/ADR cells, but has no effect on the drug sensitivities of MCF-7/VP cells that overexpress MRP1.

Product Specification

Alternative Name:N-(1-Benzyl-2,3-dihydro-1H-pyrrolo[2,3-b]quinolin-4-yl)-2-phenylacetamide
 
Formula:C26H23N3O
 
MW:393.5
 
CAS:365565-02-2
 
Purity:≥93%
 
Appearance:White to off-white powder.
 
Solubility:Soluble in methanol, 100% ethanol (3mg/ml) or DMSO (20mg/ml).
 
Shipping:Ambient
 
Long Term Storage:-20°C
 
270-290
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270-290

Product Literature References

Synthesis and evaluation of dihydropyrroloquinolines that selectively antagonize P-: B.D. Lee, et al.; J. Med. Chem. 47, 1413 (2004), Abstract;
Development of a syngeneic in vivo tumor model and its use in evaluating a novel P-glycoprotein modulator, PGP-4008: B.D. Lee, et al.; Oncol. Res. 14, 49 (2003), Abstract;

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