Online Purchasing Account You are logged on as Guest. LoginRegister a New AccountShopping cart (Empty)
United States 

Gefitinib-based PROTAC 3

VHL-recruiting PROTAC targeting on EGFR
 
ENZ-CHM261-0001 1 mg 266.00 USD
 
ENZ-CHM261-0005 5 mg 448.00 USD
 
ENZ-CHM261-0010 10 mg 700.00 USD
 
ENZ-CHM261-0025 25 mg 1,176.00 USD
 
ENZ-CHM261-0050 50 mg 1,960.00 USD
 
ENZ-CHM261-0100 100 mg 3,360.00 USD
Do you need bulk/larger quantities?
 
Gefitinib-based PROTAC 3 is targeting on EGFR, consisting of Gefitinib as the warhead linked to VHL-recruiting ligand.

Product Specification

Formula:C47H57ClFN7O8S
 
MW:934.5
 
CAS:2230821-27-7
 
Purity:≥99%
 
Appearance:White solid.
 
Solubility:Soluble in DMSO (75 mg/mL). Insoluble in water.
 
Shipping:Shipped on Blue Ice
 
Long Term Storage:-20°C
 
Regulatory Status:RUO - Research Use Only
 
ENZ-CHM261 structure
Please mouse over
ENZ-CHM261 structure

General Literature References

The Advantages of Targeted Protein Degradation Over Inhibition: An RTK Case Study: G.M. Burslem, et al.; Cell Chem. Biol. 25, 67 (2018), Abstract; Full Text

Product Toolbox

PRODUCT RESOURCES

Datasheet
MSDS
Certificate of Analysis

RELATED PRODUCTS

By target:
EGFR
Ligase [E3]
By biological activity:
EGFR Inhibitor
Ligase [E3] Ligand
By catalog section:

PRODUCT SUPPORT

FAQs
Technical Service
Customer Service

Related Literature

Catalogs
Ubiquitin & UBL Signaling Catalog
Ubiquitin & UBL Signaling Catalog
Download as PDF

All new literature pieces

Recommend this page

 
Keep in touch

©2020 Enzo Life Sciences, Inc.,