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Arv-825

PROTAC targeting on BRD4
 
ENZ-CHM258-0001 1 mg 140.00 USD
 
ENZ-CHM258-0005 5 mg 241.00 USD
 
ENZ-CHM258-0010 10 mg 371.00 USD
 
ENZ-CHM258-0025 25 mg 660.00 USD
 
ENZ-CHM258-0050 50 mg 1,124.00 USD
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ARV-825 is a PROTAC targeting on BRD4, consisting of a BRD4-ligand JQ-1 linked to a cereblon E3 ligase ligand Pomalidomide, with Kds values of 90nM and 28nM for affinity to BD1 and BD2.

Product Details

Formula:C46H47ClN8O9S
 
MW:923.4
 
CAS:1818885-28-7
 
Purity:≥98%
 
Appearance:Yellow solid.
 
Shipping:Blue Ice
 
Long Term Storage:-20°C
 
Regulatory Status:RUO - Research Use Only
 
ENZ-CHM258 structure
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ENZ-CHM258 structure

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RELATED PRODUCTS

By target:
BET bromodomain protein
Ligase [E3]
By biological activity:
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Ligase [E3] Ligand
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