Intermediate-potency protein phosphatase 2A (PP2A) inhibitor (IC50=970nM, IC50 for PP1=5000nM). Useful for structure/activity correlations. .
Product Details
| Alternative Name: | 7-Oxabicyclo[2.2.1]heptane-2,3-di-carboxylic acid |
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| Formula: | C8H10O5 |
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| MW: | 186.2 |
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| CAS: | 145-73-3 |
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| MI: | 14: 3575 |
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| Purity: | ≥98% |
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| Appearance: | White solid. |
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| Solubility: | Soluble in water (>25mg/ml). |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | Ambient |
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| Use/Stability: | Store, as supplied, at room temperature for up to 1 year. Store solutions at -20°C for up to 3 months. |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Protein phosphatase 2A and its [3H]cantharidin/[3H]endothall thioanhydride binding site. Inhibitor specificity of cantharidin and ATP analogues: Y.M. Li, et al.; Biochem. Pharmacol.
46, 1435 (1993),
Abstract;
Cantharidin-binding protein: identification as protein phosphatase 2A: Y.M. Li & J.E. Casida; PNAS
89, 11867 (1992),
Abstract;
