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Clozapine N-oxide

Major metabolite of clozapine
BML-NS105-0005 5 mg 113.00 USD
BML-NS105-0025 25 mg 462.00 USD
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  • High purity
  • Active in vitroand in vivo
  • Possesses little-to-no activity at 5-HT receptors
Clozapine N-oxide (CNO) is a major metabolite of clozapine (Prod. No. BML-D107). CNO activates designer receptors exclusively activated by designer drugs (DREADDs) that are derived from human muscarinic acetylcholine receptors (M1-5D receptors).

Product Details

Alternative Name:CNO
Formulation:Contains 1 equivalent of methanol.
Purity:≥99% (HPLC)
Appearance:Yellow solid.
Solubility:Soluble in water (5mg/ml).
Shipping:Ambient Temperature
Long Term Storage:Ambient
Scientific Background:Clozapine is an antipsychotic medication used in the treatment of schizophrenia, and is also sometimes used off-label for the treatment of bipolar disorder and borderline personality disorder. It is on the World Health Organization's List of Essential Medicines, a list of the most important medication needed in a basic health system.
Regulatory Status:RUO - Research Use Only
BML-NS105 structure
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BML-NS105 structure

Product Literature References

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