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Farnesyltransferase inhibitor
BML-G235-0001 1 mg 204.00 USD
BML-G235-0005 5 mg 746.00 USD
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A potent and selective, cell-permeable farnesyl transferase inhibitor IC50=21 nM, 30-fold selective over geranylgeranyl transferase.

Product Details

Purity:≥98% (HPLC)
Identity:Determined by ESI-MS.
Appearance:White to off-white powder.
Solubility:Soluble in DMSO (5mg/ml) or water (2mg/ml).
Shipping:Ambient Temperature
Long Term Storage:-20°C
Regulatory Status:RUO - Research Use Only
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Product Literature References

The CAAX peptidomimetic compound B581 specifically blocks farnesylated, but not geranylgeranylated or myristylated, oncogenic ras signaling and transformation: A. D. Cox, et al.; J. Biol. Chem. 269, 19203 (1994), Abstract; Full Text
Peptidomimetic inhibitors of Ras farnesylation and function in whole cells: M. A. Garcia, et al.; J. Biol. Chem. 268, 18415 (1993), Abstract; Full Text