ß-Adrenergic receptor antagonist. Serotonin 5HT1A/1B antagonist.
Product Details
Formula: | C16H21N3O2 . 1/2C4H4O4 |
|
MW: | 345.4 |
|
CAS: | 69906-85-0 |
|
Purity: | ≥99% (TLC) |
|
Appearance: | White solid. |
|
Solubility: | Soluble in warm water (2 mg/ml), DMSO (8 mg/ml). |
|
Shipping: | Ambient |
|
Long Term Storage: | Ambient |
|
Use/Stability: | Store solutions at -20°C for up to 4 months |
|
Regulatory Status: | RUO - Research Use Only |
|
Please mouse over
Product Literature References
Comparison of the profiles of agonists as stimulants of the beta 3-adrenoceptor in vitro with their gastroprotective effects in the conscious rat: A. K. Bahl, et al.; Br. J. Pharmacol.
117, 580 (1996),
Abstract;
Full Text
Characterization of 5-hydroxytryptamine receptors in goat cerebral arteries: F. J. Miranda, et al.; Gen. Pharmacol.
26, 1267 (1995),
Abstract;
Blockade of the central 5-HT autoreceptor by beta-adrenoceptor antagonists: D. N. Middlemiss, et al.; Eur. J. Pharmacol.
120, 51 (1986),
Abstract;
Cyanopindolol is a highly potent and selective antagonist at the presynaptic serotonin autoreceptor in the rat brain cortex: E. Schlicker, et al.; Naunyn. Schmied. Arch. Pharmacol.
331, 398 (1985),
Abstract;
Specificity of the beta 2-adrenergic receptor stimulating cyclic AMP accumulation in the intermediate lobe of rat pituitary gland: H. Meunier & F. Labrie ; Eur. J. Pharmacol.
81, 411 (1982),
Abstract;