A slowly dissociating β1-adrenergic receptor antagonist. Antihypertensive. Antioxidant (IC50=1.8 µM) and free radical scavenging activity.
Product Details
| Formula: | C23H28N2O3 . C3H4O4 |
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| MW: | 484.6 |
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| CAS: | 82857-38-3 |
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| Purity: | ≥97% (HPLC) |
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| Appearance: | White solid. |
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| Solubility: | Soluble in water at 3mg/ml. |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | Ambient |
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| Use/Stability: | Store solutions at -20°C for up to 4 months |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Alpha-1 and beta-adrenergic receptor blocking potencies of bopindolol and its two metabolites (18-502 and 20-785) as assessed by radioligand binding assay methods: Y. Hosohata, et al.; Gen. Pharmacol.
26, 743 (1995),
Abstract;
Antioxidative action of the beta-adrenoceptor antagonist bopindolol and its metabolite 18-502: Y. Aniya, et al.; Jpn. J. Pharmacol.
68, 323 (1995),
Abstract;
Full Text
Bopindolol is a slowly dissociating beta 1-adrenoceptor antagonist when compared to other beta-blockers: Y. Hosohata, et al.; Biol. Pharm. Bull.
18, 1066 (1995),
Abstract;
The affinity of bopindolol and its two metabolites for a beta 2-adrenoceptor in the bovine mesenteric artery: Y. Hosohata, et al.; Biol. Pharm. Bull.
17, 1296 (1994),
Abstract;
