Melatonin receptor antagonist. More potent than Luzindole (Prod. No. ALX-550-184) in the Xenopus melanophore assay.
Product Details
| Alternative Name: | N-[2-(2-Phenylindol-3-yl)ethyl] cyclobutanecarboxyamide |
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| Formula: | C21H22N2O |
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| MW: | 318.4 |
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| Purity: | ≥98% |
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| Appearance: | Oil. |
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| Solubility: | Soluble in chloroform or DMSO. |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | -20°C |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Mapping the melatonin receptor. 5. Melatonin agonists and antagonists derived from tetrahydrocyclopent[b]indoles, tetrahydrocarbazoles and hexahydrocyclohept[b]indoles: D.J. Davies, et al.; J. Med. Chem.
41, 451 (1998),
Abstract;
Mapping the melatonin receptor. 3. Design and synthesis of melatonin agonists and antagonists derived from 2-phenyltryptamines: P.J. Garratt, et al.; J. Med. Chem.
38, 1132 (1995),
Abstract;
Radioligand binding affinity and biological activity of the enantiomers of a chiral melatonin analogue: D. Sugden, et al.; Eur. J. Pharmacol.
287, 239 (1995),
Abstract;
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