Highly potent κ-opioid receptor agonist.
Product Details
Alternative Name: | 2-(3,4-Dichlorophenyl)-N-methyl-N-[(1S)-1-phenyl-2-(1-pyrrolidinyl)ethyl]acetamide . HCl |
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Formula: | C21H24Cl2N2O . HCl |
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MW: | 427.8 |
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CAS: | 115199-84-3 |
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Appearance: | White solid. |
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Solubility: | Soluble in methanol or 100% ethanol. |
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Shipping: | Ambient |
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Long Term Storage: | +4°C |
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Handling: | Protect from light. |
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Regulatory Status: | RUO - Research Use Only |
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Product Literature References
2-(3,4-Dichlorophenyl)-N-methyl-N-[2-(1-pyrrolidinyl)-1-substituted- ethyl]-acetamides: the use of conformational analysis in the development of a novel series of potent opioid kappa agonists: G.F. Costello, et al.; J. Med. Chem.
34, 181 (1991),
Abstract;
Structure/activity studies related to 2-(3,4-dichlorophenyl)-N-methyl-N-[2-(1-pyrrolidinyl)-1-substituted-ethyl]acetamides: a novel series of potent and selective kappa-opioid agonists: J.J. Barlow, et al.; J. Med. Chem.
34, 3149 (1991),
Abstract;