Inhibits calmodulin stimulation of cyclic nucleotide phosphodiesterase. Dopamine antagonist. D2 antagonist. H1 antagonist. Inhibits TNF-α production. Potent PLA2 inhibitor. Inhibits nitric oxide synthase (NOS) in mouse brain and prevents lipopolysaccharide induction of NOS in mouse lung. Antipsychotic.
Product Details
| Alternative Name: | 2-Chloro-10-(3-dimethylaminopropyl)phenothiazine . HCl |
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| Formula: | C17H19ClN2S . HCl |
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| MW: | 355.3 |
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| CAS: | 69-09-0 |
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| MI: | 14: 2185 |
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| RTECS: | SO1750000 |
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| Purity: | ≥98% (UHPLC) |
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| Appearance: | White to off-white powder. |
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| Solubility: | Soluble in 100% ethanol, methanol or water (50mg/ml). |
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| Shipping: | Ambient Temperature - Dangerous Good |
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| Long Term Storage: | Ambient |
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| Use/Stability: | Not stable in aqueous solution. We strongly recommend always to use freshly prepared solutions. |
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| Handling: | Protect from light. |
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| Regulatory Status: | RUO - Research Use Only |
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