Selective ETA antagonist.
Product Details
| Sequence: | (Hexahydro-1H-azepinyl)carbonyl-Leu-D-Trp(Me)-D-Ala(2-pyridyl)-OH |
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| Formula: | C32H43N6O5 |
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| MW: | 605.8 |
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| Quantity: | *Sold as net peptide weight. |
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| Purity: | ≥97% |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | -20°C |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Effect of different endothelin receptor antagonists and of the novel non-peptide antagonist Ro 46-2005 on endothelin levels in rat plasma: B.-M. Löffler, et al.; FEBS Lett.
333, 108 (1993),
Abstract;
Structure-activity relationships of C-terminal endothelin hexapeptide antagonists: A.M. Doherty, et al.; J. Med. Chem.
36, 2585 (1993),
Abstract;
