Very potent ETA antagonist.
Product Details
Sequence: | cyclo(D-Asp-Pro-D-Ile-Leu-D-Trp) |
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Formula: | C32H44N6O7 |
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MW: | 624.7 |
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Quantity: | *Sold as net peptide weight. |
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Purity: | ≥96% |
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Appearance: | White to off-white lyophilized powder. |
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Solubility: | 1mg/ml completely soluble in 5% acetic acid. |
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Shipping: | Ambient |
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Long Term Storage: | -20°C |
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Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Characterization of [125I]-endothelin-1 and [125I]-BQ3020 binding to rat cerebellar endothelin receptors: P.S. Widdowson & C.N. Kirk; Br. J. Pharmacol.
118, 2126 (1996),
Abstract;
The endothelin receptor profile in L6 myotubes: Z. Fekete, et al.; Pharmacol. Exp. Ther.
275, 215 (1995),
Abstract;
Lippton et al. ; American Heart Association, 66th Scientific Sessions, Georgia (World Congress, Nov. 8-11, 1993) 66, 8 (1993),