Replaces Prod. #: ALX-270-075
KT5720 is a hexylester derivative of K-252a and is a selective inhibitor of PKA (Ki=0.056 µM). Cell permeable.
Product Details
| Formula: | C32H31N3O5 |
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| MW: | 537.6 |
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| CAS: | 108068-98-0 |
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| Purity: | ≥98% (HPLC) |
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| Appearance: | White powder. |
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| Solubility: | Soluble in methanol: clear colorless solution at 5mg/ml. |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | -20°C |
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| Use/Stability: | Stable for at least 1 year after receipt when stored, as supplied, at -20°C. Stock solutions are stable for up to 3 months at -20°C. |
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| Handling: | Protect from light. |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Effects of insulin, insulin-like growth factor-I, and phorbol esters on neutral cholesteryl esterase activity in cultured rat vascular smooth muscle cells.: R. Fujiwara, et al.; J. Lab. Clin. Med.
126, 240 (1995),
Abstract;
Effects of selective inhibition of protein kinase C, cyclic AMP-dependent protein kinase, and Ca(2+)-calmodulin-dependent protein kinase on neurite development in cultured rat hippocampal neurons: L. Cabell & G. Audesirk; Int. J. Dev. Neurosci.
11, 357 (1993),
Abstract;
Multiple kinase arrest points in the G1 phase of nontransformed mammalian cells are absent in transformed cells.: D.M. Gadbois, et al.; Proc. Natl. Acad. Sci. USA
89, 8626 (1992),
Abstract;
K-252 compounds, novel and potent inhibitors of protein kinase C and cyclic nucleotide-dependent protein kinases: H. Kase, et al.; Biochem. Biophys. Res. Commun.
142, 436 (1987),
Abstract;
