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SB-366791

TRPV1 antagonist
 
BML-VR105-0005 5 mg 68.00 USD
 
BML-VR105-0025 25 mg 279.00 USD
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Replaces Prod. #: ALX-550-388

A potent and selective vanilloid receptor (TRPV1) antagonist. An effective antagonist of hTRPV1 when stimulated by capsaicin, acid, or noxious heat.

Product Specification

Formula:C16H14NO2Cl
 
MW:287.8
 
CAS:472981-92-3
 
Purity:≥98% (TLC)
 
Appearance:Beige solid.
 
MeltingPoint:165-167°C
 
Solubility:Soluble in DMSO (25mg/ml) or 100% ethanol (10mg/ml with warming).
 
Shipping:Ambient
 
Long Term Storage:Ambient
 
Use/Stability:Store, as supplied, at room temperature for up to 1 year. Store solutions at -20°C for up to 3 months.
 
BML-VR105 structure
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BML-VR105 structure

Product Literature References

TRPV1, ASICs and P2X2/3 expressed in bone cells simultaneously regulate bone metabolic markers in ovariectomized mice: K. Kanaya, et al.; J. Musculolskelet. Neuronal Interact. 16, 145 (2016), Abstract;
Effects of the novel TRPV1 receptor antagonist SB366791 in vitro and in vivo in the rat: A. Varga, et al.; Neurosci. Lett. 385, 137 (2005), Abstract;
Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist: M.J. Gunthorpe, et al.; Neuropharmacology 46, 133 (2004), Abstract;
Identification of SB-366791, a potent and selective antagonist of vanilloid receptor-1: H.K. Rami, et al.; Drugs Fut. 27 (Supply A), 411 (2002),

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