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TRPV1 agonist
BML-VR102-0025 25 mg 228.00 USD
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Replaces Prod. #: ALX-550-398

Endogenous TRPV1 agonist (Ki=36nM, EC50=36nM) with weak affinity for rat CB1 receptor (Ki=1.6µM). Potent inhibitor of 5-lipoxygenase (IC50=7.5nM) and of early and late events in TCR mediated T cell activation. Inhibits NF-κB dependent transcriptional activity without affecting either degradation of the cytoplasmic NF-κB inhibitory protein, IκBα, or DNA binding activity.

Product Specification

Alternative Name:OLDA, N-[2-(3,4-Dihydroxyphenyl)ethyl]-9Z-octadecenamide
Purity:≥98% (TLC)
Appearance:White solid.
Solubility:Soluble in DMSO (20mg/ml).
Shipping:Shipped on Dry Ice
Long Term Storage:-20°C
Use/Stability:Stable for at least 1 year after receipt when stored at -20°C. We do not recommend storing aqueous solutions for more than one day.
Handling:Protect from light.
BML-VR102 structure
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BML-VR102 structure

Product Literature References

Direct evidence for activation and desensitization of the capsaicin receptor by N-oleoyldopamine on TRPV1-transfected cell, line in gene deleted mice and in the rat: J. Szolcsanyi, et al.; Neurosci. Lett. 361, 155 (2004), Abstract;
Immunosuppressive activity of endovanilloids: N-arachidonoyl-dopamine inhibits activation of the NF-kappa B, NFAT, and activator protein 1 signaling pathways: R. Sancho, et al.; J. Immunol. 172, 2341 (2004), Abstract;
N-oleoyldopamine, a novel endogenous capsaicin-like lipid that produces hyperalgesia: C.J. Chu, et al.; J. Biol. Chem. 278, 13633 (2003), Abstract;
Inhibition of in vitro prostaglandin and leukotriene biosyntheses by cinnamoyl-beta-phenethylamine and N-acyldopamine derivatives: C.F. Tseng, et al.; Chem. Pharm. Bull. 40, 396 (1992), Abstract;
Inhibition of arachidonate 5-lipoxygenase by phenolic compounds: S. Iwakami, et al.; Chem. Pharm. Bull. 34, 3960 (1986), Abstract;

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