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BML-288

PDE2 inhibitor
 
BML-PD200-0005 5 mg 69.00 USD
 
BML-PD200-0025 25 mg 303.00 USD
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Potent (IC50=40nM) and selective (290X selectivity over other PDE isoforms) inhibitor of phosphodiesterase Type II (PDE2). Displayed no significant level of binding to neither a collection of 54 receptors and ion channels, nor to a panel of 30 kinases. BML-288 demonstrated no inhibition of 5-lipoxygenase (5-LO) or cyclooxygenase (COX-1). BML-288 is more potent and selective than EHNA (BML-PD129).

Product Specification

Alternative Name:5-Methyl-6-oxo-N-(1,3,4-thiadiazol-2-yl)-7H-furo[2,3-f]indole-7-carboxamide
 
Formula:C14H10N4O3S
 
MW:314.3
 
Purity:≥98% (TLC)
 
Appearance:Off-white solid.
 
MeltingPoint:243-245°C
 
Solubility:Soluble in DMSO (25 mg/ml).
 
Shipping:Shipped on Blue Ice
 
Long Term Storage:-20°C
 
Use/Stability:Store under inert gas.  Compound will darken on exposure to air.  Stable for at least 1 year after the date of reciept when stored at -20°C. Solutions can be stored at -20°C for up to 3 months.
 
Handling:Solutions can be stored at -20°C for up to 3 months.
 
BML-PD200 Structure
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BML-PD200 Structure

Product Literature References

A new chemical tool for exploring the physiological function of the PDE2 isozyme: R. Chambers, et al.; Bioorg. Med. Chem. Lett. 16, 307 (2006), Abstract;

Related Products

EHNA 

PDE inhibitor
51350-19-7, ≥98% (HPLC) | Print as PDF
 
BML-PD129-0010 10 mg 61.00 USD
 
BML-PD129-0050 50 mg 240.00 USD
Do you need bulk/larger quantities?
 

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