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Nalmefene . HCl

Opioid receptor inhibitor
 
BML-NO110-0500 500 mg 357.00 USD
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Opioid receptor antagonist similar to naloxone but with a slower onset and longer duration of action. Antagonizes the effects of salvinorin (κ-agonist) as well as herkinorin (µ-agonist). A promising drug for the treatment of alcohol dependence.

Product Specification

Alternative Name:(5α)-17-(Cyclopropylmethyl)-4,5-epoxy-6-methylene-morphinan-3,14-diol
 
Formula:C21H25NO3 . HCl
 
MW:339.4 . 36.5
 
CAS:58895-64-0
 
Purity:≥99% (TLC)
 
Appearance:White solid.
 
Solubility:Soluble in water (>25mg/ml).
 
Shipping:Ambient
 
Long Term Storage:Ambient
 
Use/Stability:Store solutions at -20°C for up to 3 months.
 
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Product Literature References

In vivo characterization of the opioid antagonist nalmefene in mice: M.D. Osborn, et al.; Life Sci. 86, 624 (2010), Abstract;
Unconditioned behavioral effects of the powerful kappa-opioid hallucinogen salvinorin A in nonhuman primates: fast onset and entry into cerebrospinal fluid: E.R. Butelman, et al.; J. Pharmacol. Exp. Ther. 328, 588 (2009), Abstract;
Opioid antagonists for pharmacological treatment of alcohol dependence - a critical review: M. Soyka & S. Rosner; Curr. Drug Abuse Rev. 1, 280 (2008), Abstract;
The effects of herkinorin, the first mu-selective ligand from a salvinorin A-derived scaffold, in a neuroendocrine biomarker assay in nonhuman primates: E.R. Butelman, et al.; J. Pharmacol. Exp. Ther. 327, 154 (2008), Abstract;

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