SCH-202676

Blocks agonist and antagonist binding to G protein-coupled receptors



BML-G521-0010	10 mg	100.00 USD

BML-G521-0050	50 mg	403.00 USD

Modulator of both agonist and antagonist binding to G protein-coupled receptors which functions via thiol modification rather than true allosteric mechanisms. Has been shown to block agonist or antagonist activity at adenosine, adrenergic, dopaminergic, muscarinic, opioid and P2Y. IC₅₀s vary from 0.1 to 1.8µM.The nature of the interaction of SCH-202676 and receptors is dependent on whether it is studied using intact versus broken cell preparations.

Product Specification

Formula:	C₁₅H₁₃N₃S . HBr

MW:	348.3

Purity:	≥99% (HPLC)

Appearance:	Yellow solid.

CAS:	70375-43-8

Solubility:	Soluble in DMSO (7mg/ml, with warming).

Long Term Storage:	Ambient

Background / Technical Information:	Please click here for the comprehensive product data sheet.