URB-597

FAAH inhibitor



BML-EI327-0005	5 mg	37.00 USD

BML-EI327-0025	25 mg	151.00 USD

Replaces Prod. #: ALX-550-382

URB-597 is a potent and selective inhibitor of the enzyme fatty acid amide hydrolase (FAAH), which is involved in the hydrolysis of endogenous cannabinoids such as anandamide. Inhibition of FAAH may serve to enhance the analgesic effects of endogenous cannabinoids. URB-597 has been shown to inhibit FAAH in rat cortical neuron membranes and in intact neurons with IC₅₀values of 4.6nM and 0.5nM, respectively. The compound has also been shown to have anxiolytic effects in rats (ID₅₀=0.15mg/kg).

Formula:	C₂₀H₂₂N₂O₃

Purity:	≥98% (TLC)

Appearance:	White solid.

CAS:	546141-08-6

Solubility:	Soluble in 100% ethanol (1mg/ml), dimethyl formamide (10mg/ml) or DMSO (10mg/ml)

Long Term Storage:	-20°C

Use/Stability:	Store, as supplied, at -20°C for up to 1 year. Store solutons at -20°C for up to 3 months.

Hazard:	DANGEROUS FOR THE ENVIRONMENT TOXIC.

Handling:	Protect from light.

Background / Technical Information:	Please click here for the comprehensive product datasheet.