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AG-825

EGFR inhibitor
 
BML-EI267-0002 2 mg 86.00 USD
 
BML-EI267-0010 10 mg 325.00 USD
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Replaces Prod. #: ALX-270-137

A selective HER1-2 (HER2-Neu) tyrosine kinase inhibitor (IC50 = 0.35µM vs. 19µM for EGFR and 40µM for PDGFR). Not active in whole cells due to high intracellular ATP concentrations.

Product Specification

Alternative Name:Tyrphostin AG 825, Tyrphostin C15, 5-[(Benzothiazol-2-yl)thiomethyl]-4-hydroxy-3-methoxybenzyl-idenecyanoacetamide
 
Formula:C19H15N3O3S2
 
MW:397.5
 
CAS:149092-50-2
 
Purity:≥98% (TLC)
 
Appearance:Yellow solid.
 
Solubility:Soluble in DMSO (25mg/ml) or methanol.
 
Shipping:Ambient
 
Long Term Storage:Ambient
 
Use/Stability:Stable for at least 1 year after receipt when stored at +20°C. Stock solutions are stable for up to 3 months at -20°C.
 
Handling:Protect from light.
 
Technical Info/Product Notes:Note: Product is not sterile.
 
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Product Literature References

Tyrosine kinase inhibition: an approach to drug development: A. Levitzki & A. Gazit; Science 267, 1782 (1995), Abstract;
Selective inhibition of the epidermal growth factor and HER2/neu receptors by tyrphostins: N. Osherov, et al.; J. Biol. Chem. 268, 11134 (1993), Abstract;

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