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CCR8 activator
BML-CX101-0010 10 mg 107.00 USD
BML-CX101-0050 50 mg 443.00 USD
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Novel small molecule agonist at the CCR8 chemokine receptor (EC50=254nM) with no activity at CCR1, CCR2B, CCR4, CCR5, CXCR2, CXCR3 or CXCR4. Dose dependently increases intracellular calcium and stimulates extracellular acidification in cells expressing human CCR8. Murine CCR8-expressing cells underwent chemotaxis on exposure to this agonist. Inhibits HIV fusion of cells expressing CD4 and CCR8. Small molecule CCR8 agonists represent useful tools for exploring CCR8 biology especially in experiments where the use of the natural protein agonist is impractical.

Product Specification

Alternative Name:2-[2-[4-[(3-Phenoxyphenyl)methyl]-1-piperazinyl]ethoxy]ethanol dihydrochloride
Formula:C21H28N2O3 . 2HCl
MW:356.4 . 73.0
Purity:≥98% (TLC)
Appearance:White solid.
Solubility:Soluble in water (5 mg/ml) or DMSO (4 mg/ml).
Long Term Storage:Ambient
Use/Stability:Store, as supplied, at room temperature for up to one year.  Store solutions at -20°C for up to 3 months.
BML-CX101 Structure
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BML-CX101 Structure

Product Literature References

Molecular interaction of a potent nonpeptide agonist with the chemokine receptor CCR8.: P.A. Jensen, et al.; Mol. Pharmacol. 72, 327 (2007), Abstract;
Identification and Characterization of a Potent, Selective Nonpeptide Agonist of the CC Chemokine Receptor CCR8 : C.A. Haskell, et al. ; Mol. Pharmacol. 69, 309 (2006), Abstract; Full Text

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