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PSY-279

TRPV1 agonist
 
ALX-550-397-M005 5 mg 218.00 USD
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TRPV1 agonist. Amide based RTX analog. RTX binding affinity (Ki=15nM), high agonism (calcium influx: EC50=0.29nM).

Product Specification

Alternative Name:N-[2-(4-tert-Butylbenzyl)-3-(pivaloylxy)propyl]-2-[4-hydroxy-3-methoxyphenyl]acetamide
 
Formula:C28H39NO5
 
MW:469.6
 
CAS:289903-41-9
 
Purity:≥98%
 
Appearance:White sticky solid.
 
Solubility:Soluble in methanol, 100% ethanol, DMSO or other organic solvents; insoluble in water.
 
Shipping:Ambient
 
Long Term Storage:-20°C
 
Handling:Protect from light.
 
550-397
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550-397

Product Literature References

Structure-activity relationships of simplified resiniferatoxin analogues with potent VR1 agonism elucidates an active conformation of RTX for VR1 binding: J. Lee, et al.; Bioorg. Med. Chem. 12, 1055 (2004), Abstract;
Phenolic modification as an approach to improve the pharmacology of the 3-acyloxy-2-benzylpropyl homovanillic amides and thioureas, a promising class of vanilloid receptor agonists and analgesics: J. Lee, et al.; Bioorg. Med. Chem. 10, 1171 (2002), Abstract;

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