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8-(4-Chlorophenylthio)guanosine 3',5'-cyclic Monophosphothioate, Rp-Isomer . triethylammonium salt (high purity)

PKG inhibitor
 
ALX-480-032-C100 100 µg 61.00 USD
 
ALX-480-032-M001 1 mg 289.00 USD
Do you need bulk/larger quantities?
 
Potent selective inhibitor of cGMP-dependent protein kinase 1α, 1β and type II. Resistant to mammalian cyclic nucleotide-dependent phosphodiesterases, no metabolic side effects. Significantly more lipophilic and membrane permeant as compared to Rp-cGMPS (Prod. No. ALX-480-072) or Rp-8-Br-cGMPS (Prod. No. BML-CN216).

Product Specification

Alternative Name:Rp-8-pCPT-cGMPS . TEA, 8-pCPT-cGMPS . TEA, Rp-Isomer
 
Formula:C16H14ClN5O6PS2 . C6H16N
 
MW:502.9 . 102.2
 
CAS:153660-04-9
 
Purity:≥99% (HPLC)
 
Identity:Determined by UV and ESI-MS.
 
Appearance:White to off-white crystalline powder.
 
Solubility:Soluble in water and aqueous buffers.
 
Shipping:Ambient
 
Long Term Storage:-20°C
 
ALX-480-032
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ALX-480-032

Product Literature References

Green tea catechins enhance norepinephrine-induced lipolysis via a protein kinase A-dependent pathway in adipocytes: S. Chen, et al.; Biochem. Biophys. Res. Commun. 461, 1 (2015), Application(s): Cell Culture, Abstract;
Antagonists of cyclic nucleotide-gated channels and molecular mapping of their site of action: R.H. Kramer & G.R. Tibbs; J. Neurosci. 16, 1285 (1996), Abstract;
The type II isoform of cGMP-dependent protein kinase is dimeric and possesses regulatory and catalytic properties distinct from the type I isoforms: D.M. Gamm, et al.; J. Biol. Chem. 270, 27380 (1995), Abstract; Full Text
(Rp)-8-pCPT-cGMPS, a novel cGMP-dependent protein kinase inhibitor: E. Butt, et al.; Eur. J. Pharmacol. 269, 265 (1994), Abstract;

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Guanosine 3',5'-cyclic Monophosphothioate, Rp-Isomer . sodium salt 

PKG inhibitor
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Rp-8-Br-cGMPS 

PKG inhibitor
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