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Thiocolchicoside

GABAA receptor antagonist
 
ALX-350-374-M005 5 mg 125.00 USD
 
ALX-350-374-M025 25 mg 478.00 USD
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Potent competitive antagonist of GABAAR function. Muscle relaxant. Displays anti-inflammatory and analgesic properties. Shows strong epileptogenic and convulsant activity.

Product Specification

Alternative Name:2-Demethoxy-2-glucosidoxythiocolchicine
 
Formula:C27H33NO10S
 
MW:563.6
 
Source:Semisynthetic.
 
CAS:602-41-5
 
MI:14: 9324
 
Purity:≥95% (HPLC)
 
Identity:Identity determined by 1H-NMR.
 
Appearance:Yellow solid.
 
Solubility:Soluble in water or 100% ethanol.
 
Shipping:Ambient
 
Long Term Storage:-20°C
 
350-374
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350-374

Product Literature References

Thiocolchicoside inhibits the activity of various subtypes of recombinant GABA(A) receptors expressed in Xenopus laevis oocytes: M.P. Mascia, et al.; Eur. J. Pharmacol. 558, 37 (2007), Abstract;
The muscle relaxant thiocolchicoside is an antagonist of GABAA receptor function in the central nervous system: M. Carta, et al.; Neuropharmacology 51, 805 (2006), Abstract;
Focal and secondarily generalised convulsive status epilepticus induced by thiocolchicoside in the rat: G. Sechi, et al.; Seizure 12, 508 (2003), Abstract;
Review of the toxicology, pharmacodynamics and pharmacokineticss of thiocolchicoside, a GABA-agonist muscle relaxant with anti-inflammatory and analgesic actions: J.M. Janbroers; Acta Ther. 13, 221 (1987),

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