Selective high affinity inhibitor of P-glycoprotein (MDR1).
Product Details
| Alternative Name: | Boc-Asp(OBzl)-Lys(Z)-OtBu |
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| Formula: | C34H47N3O9 |
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| MW: | 641.8 |
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| Purity: | ≥98% (HPLC) |
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| Appearance: | White to off-white powder. |
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| Solubility: | Soluble in DMSO. |
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| Shipping: | Ambient Temperature |
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| Long Term Storage: | -20°C |
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| Regulatory Status: | RUO - Research Use Only |
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Product Literature References
Insights into the structure and substrate interactions of the P- glycoprotein multidrug transporter from spectroscopic studies: F.J. Sharom, et al.; Biochim. Biophys. Acta
1461, 327 (1999),
Abstract;
Interaction of the P-glycoprotein multidrug transporter (MDR1) with high affinity peptide chemosensitizers in isolated membranes, reconstituted systems, and intact cells: F.J. Sharom, et al.; Biochem. Pharmacol.
58, 571 (1999),
Abstract;
Micellar electrokinetic chromatography of highly hydrophobic peptides: M. Idei, et al.; Anal. Chim. Acta 372, 273 (1998),
