ET_A receptor antagonist [FR 139317]



ALX-155-017-PC05	0.5 mg*	117.00 USD

ALX-155-017-P001	1 mg*	221.00 USD

Selective ET_Aantagonist.

Product Specification

Formula:	C₃₂H₄₃N₆O₅

MW:	605.8

Quantity:	*Sold as net peptide weight.

Purity:	≥97%

Sequence:	(Hexahydro-1H-azepinyl)carbonyl-Leu-D-Trp(Me)-D-Ala(2-pyridyl)-OH

Long Term Storage:	-20°C

Product Literature References

Effect of different endothelin receptor antagonists and of the novel non-peptide antagonist Ro 46-2005 on endothelin levels in rat plasma: B.-M. Löffler, et al.; FEBS Lett. 333, 108 (1993), Abstract;

Structure-activity relationships of C-terminal endothelin hexapeptide antagonists: A.M. Doherty, et al.; J. Med. Chem. 36, 2585 (1993), Abstract;