ET_B receptor agonist [BQ-3020]



ALX-155-015-PC05	0.5 mg*	83.00 USD

Selective ligand for the ET_Breceptor.

Product Specification

Alternative Name:	N-Acetyl-[Ala^11,15]-Endothelin-1

Formula:	C₉₆H₁₄₀N₂₀O₂₅S

MW:	2006.3

Quantity:	*Sold as net peptide weight.

Purity:	≥97%

Sequence:	Ac-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp-OH

Long Term Storage:	-20°C

Product Literature References

Identification of a ligand-binding site of the human endothelin-A receptor and specific regions required for ligand selectivity: M. Adachi, et al.; Eur. J. Biochem. 220, 37 (1994), Abstract;

Distinct subdomains of human endothelin receptors determine their selectivity to endothelinA-selective antagonist and endothelinB- selective agonists: A. Sakamoto, et al.; J. Biol. Chem. 268, 8547 (1993), Abstract; Full Text

A novel radioligand [125I]BQ-3020 selective for endothelin (ETB) receptors: M. Ihara, et al.; Life Sci. 51, PL47 (1992), Abstract;